| Metric | >=75kg patients N = 971 |
<75kg patients N = 1031 |
|---|---|---|
| Day 1 | ||
| AUC (ng/mL*h) | 122 (98–154) | 144 (120–174) |
| Cmax (ng/mL) | 10.17 (7.47–12.80) | 10.26 (8.23–13.42) |
| tmax (h) | 2.00 (1.00–6.00) | 2.00 (1.00–6.00) |
| Ctrough (ng/mL) | 2.24 (1.25–3.90) | 3.46 (2.20–4.60) |
| Day 7 | ||
| AUC (ng/mL*h) | 168 (121–236) | 233 (164–305) |
| Cmax (ng/mL) | 13.4 (9.9–18.4) | 16.4 (12.6–21.1) |
| tmax (h) | 2.00 (1.00–6.00) | 2.00 (1.00–6.00) |
| Ctrough (ng/mL) | 3.23 (1.27–5.85) | 5.95 (3.03–9.21) |
| 1 Median (5% Centile–95% Centile) | ||